Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2120 |
I-BET151
GSK1210151A |
Epigenetic Reader Domain | Chromatin/Epigenetic |
I-BET151 (GSK1210151A) 是 BRD2/3/4 的特异性 BET 抑制剂,IC50值分别为0.5、0.25、0.79 μM。 | |||
T22845 |
I-BET151 dihydrochloride
I-BET 151 hydrochloride |
Others | Others |
I-BET 151 dihydrochloride is a BET bromodomain inhibitor that prevents BET from recruiting to chromatin. |